Synthesis, In Vitro Biological Evaluation and Molecular Modeling of Benzimidazole-Based Pyrrole/Piperidine Hybrids Derivatives as Potential Anti-Alzheimer Agents
Benzimidazole-based pyrrole/piperidine analogs (1–26) were synthesized and then screened for their acetylcholinesterase and butyrylcholinesterase activities. All the analogs showed good to moderate cholinesterase activities. Synthesized compounds (1–13) were screened in cholinesterase enzyme inhibit...
الحاوية / القاعدة: | Pharmaceuticals |
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المؤلف الرئيسي: | |
التنسيق: | مقال |
اللغة: | English |
منشور في: |
Multidisciplinary Digital Publishing Institute (MDPI)
2024
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الوصول للمادة أونلاين: | https://www.scopus.com/inward/record.uri?eid=2-s2.0-85191352219&doi=10.3390%2fph17040410&partnerID=40&md5=09d4ff1950e1e6bbb3f21b4c293d4720 |