Synthesis, In Vitro Biological Evaluation and Molecular Modeling of Benzimidazole-Based Pyrrole/Piperidine Hybrids Derivatives as Potential Anti-Alzheimer Agents

Benzimidazole-based pyrrole/piperidine analogs (1–26) were synthesized and then screened for their acetylcholinesterase and butyrylcholinesterase activities. All the analogs showed good to moderate cholinesterase activities. Synthesized compounds (1–13) were screened in cholinesterase enzyme inhibit...

وصف كامل

التفاصيل البيبلوغرافية
الحاوية / القاعدة:Pharmaceuticals
المؤلف الرئيسي: 2-s2.0-85191352219
التنسيق: مقال
اللغة:English
منشور في: Multidisciplinary Digital Publishing Institute (MDPI) 2024
الوصول للمادة أونلاين:https://www.scopus.com/inward/record.uri?eid=2-s2.0-85191352219&doi=10.3390%2fph17040410&partnerID=40&md5=09d4ff1950e1e6bbb3f21b4c293d4720